Target & Activity
| Target | Activity | Value |
|---|---|---|
| mAChR3 | Ki | 15 nM |
| mAChR1 | Ki | 28 nM |
| mAChR2 | Ki | 260 nM |
Fig. 1 · Structure
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YM-58790
M3 muscarinic receptor antagonist
YM-58790 is a potent antagonist of M3 muscarinic receptor, with Ki of 15 nM.
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Biological Activity
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 214558-72-2 |
| Applications | M3 muscarinic receptor antagonist |
| Formula | C27H32ClN3O2 |
| Molecular Weight | 466.01 |
| SMILES | O=C(OC1CCN(CC2=CC=C(NC)C=C2)CC1)NC(C3=CC=CC=C3)C4=CC=CC=C4.[H]Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.