Fig. 1 · Structure
Documents & Downloads
YM471 free base
Cat. No.
A73184
CAS
183173-00-4
Endogenous Metabolite
YM471 free base is a selective non-peptide antagonist targeting vasopressin V1A and V2 receptors. It demonstrates high affinity for these receptors in rat models, with binding affinities (K values) of 0.16 nM for V1A and 0.77 nM for V2. This compound is valuable for investigating the role of vasopressin receptors in various physiological and pathological conditions.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 183173-00-4 |
| Applications | Endogenous Metabolite |
| Formula | C39H38F2N4O3 |
| Molecular Weight | 648.74 |
| SMILES | O=C(C1=CC=C(C=C1)NC(C2=C(C3=CC=CC=C3)C=CC=C2)=O)N4C5=CC=CC=C5/C(C(F)(CC4)F)=C/C(N6CCC(CC6)N(C)C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.