Biological Activity
Cenerimod (ACT-334441) is a potent and orally available sphingosine 1-phosphate 1 receptor (S1P1) agonist extracted from patent WO 2016184939 A1 and WO 2011007324 A1, example 1, with an EC50 of 2.7 nM.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.05 mL | 110.25 mL | 220.49 mL |
0.5 mM | 4.41 mL | 22.05 mL | 44.1 mL |
1 mM | 2.2 mL | 11.02 mL | 22.05 mL |
5 mM | 0.44 mL | 2.2 mL | 4.41 mL |
*The above data is based on the productmolecular weight 453.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A20913 |
---|---|
Actions | Agonist |
CAS No. | 1262414-04-9 |
Formula | C25H31N3O5 |
M. Wt | 453.53 |
Purity | >98% |
Synonyms | ACT-334441, ACT 334441, ACT334441 |
SMILES | OC[[email protected]](O)COC1=C(C)C=C(C2=NOC(C3=CC(C4CCCC4)=NC(OC)=C3)=N2)C=C1CC |
Storage | Store lyophilized at -20ºC, keep desiccated. |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy Cenerimod | Cenerimod Supplier | purchase | cost | manufacturer | order | distributor | buy 1262414-04-9| 1262414-04-9 Supplier | purchase 1262414-04-9 | 1262414-04-9 cost | 1262414-04-9 manufacturer | order 1262414-04-9 | 1262414-04-9 distributor