Cinanserin is a potent and selective antagonist of the 5-HT2 receptor, exhibiting Ki values of 41 nM for 5-HT2 and 3500 nM for the 5-HT1 receptor. Additionally, it acts as an inhibitor of the SARS-CoV 3CLpro, demonstrating KD values of 49.4 µM and 18.2 µM against SARS-CoV 3CLpro and HCoV-229E 3CLpro, respectively. Cinanserin has been shown to effectively reduce systemic burn edema levels, making it valuable for research in neuropharmacology and viral pathogenesis.
Cinanserin is a potent and selective antagonist of the 5-HT2 receptor, exhibiting Ki values of 41 nM for 5-HT2 and 3500 nM for the 5-HT1 receptor. Additionally, it acts as an inhibitor of the SARS-CoV 3CLpro, demonstrating KD values of 49.4 µM and 18.2 µM against SARS-CoV 3CLpro and HCoV-229E 3CLpro, respectively. Cinanserin has been shown to effectively reduce systemic burn edema levels, making it valuable for research in neuropharmacology and viral pathogenesis.
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