CSV0C018875 hydrochloride is a selective inhibitor of G9a (EHMT2), effectively blocking its enzymatic activity in both enzyme and cell-based assays. This compound demonstrates a lower toxicity profile compared to the known G9a inhibitor BIX-01294, making it a valuable tool for research. CSV0C018875 binds tightly to the active site of G9a, enhancing the compound's inhibitory potency and prolonging its residence time. Its potential for improved ADME (absorption, distribution, metabolism, and excretion) and pharmacodynamic properties positions CSV0C018875 as a promising candidate for further biological studies.
CSV0C018875 hydrochloride is a selective inhibitor of G9a (EHMT2), effectively blocking its enzymatic activity in both enzyme and cell-based assays. This compound demonstrates a lower toxicity profile compared to the known G9a inhibitor BIX-01294, making it a valuable tool for research. CSV0C018875 binds tightly to the active site of G9a, enhancing the compound's inhibitory potency and prolonging its residence time. Its potential for improved ADME (absorption, distribution, metabolism, and excretion) and pharmacodynamic properties positions CSV0C018875 as a promising candidate for further biological studies.
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