DDR1-IN-1

Catalog No.: A13985

DDR1 receptor inhibitor

DDR1-IN-1

DDR1-IN-1 Chemical Structure

CAS NO. 1449685-96-4

DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with IC50/EC50 of 105 nM/87 nM, 4-fold less potent for DDR2 (IC50= 413 nM).

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$125.00
25 mg
$250.00
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Biological Activity

DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with IC50/EC50 of 105 nM/87 nM, 4-fold less potent for DDR2 (IC50= 413 nM).
Targets
DDR1 DDR2
105 nM413 nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.1 mL 90.48 mL 180.97 mL
0.5 mM 3.62 mL 18.1 mL 36.19 mL
1 mM 1.81 mL 9.05 mL 18.1 mL
5 mM 0.36 mL 1.81 mL 3.62 mL

*The above data is based on the productmolecular weight 552.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13985
Actions Inhibitor
M. Wt 552.59
Formula C30H31F3N4O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1449685-96-4
SMILES CCN1CCN(CC1)CC2=C(C=C(C=C2)C(=O)NC3=CC(=C(C=C3)C)OC4=CC5=C(C=C4)NC(=O)C5)C(F)(F)F

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