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DDR1-IN-1 is a potent and selective DDR1 receptor tyrosine kinase inhibitor with IC50/EC50 of 105 nM/87 nM, 4-fold less potent for DDR2 (IC50= 413 nM).
Targets
| DDR1 | DDR2 | |||
| 105 nM | 413 nM |
| In vitro | DMSO | Warmed: 87 mg/mL (157.44 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 3 mg/mL (5.42 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 18.1 mL | 90.48 mL | 180.97 mL |
| 0.5 mM | 3.62 mL | 18.1 mL | 36.19 mL |
| 1 mM | 1.81 mL | 9.05 mL | 18.1 mL |
| 5 mM | 0.36 mL | 1.81 mL | 3.62 mL |
*The above data is based on the productmolecular weight 552.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A13985 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1449685-96-4 |
| Formula | C30H31F3N4O3 |
| M. Wt | 552.59 |
| Purity | >98% |
| SMILES | CCN1CCN(CC1)CC2=C(C=C(C=C2)C(=O)NC3=CC(=C(C=C3)C)OC4=CC5=C(C=C4)NC(=O)C5)C(F)(F)F |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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