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DprE1-IN-8

DprE1 Inhibitor

DprE1-IN-8 is a potent inhibitor of DprE1, demonstrating an IC50 value of less than 0.75 μM. This compound shows remarkable efficacy against Mycobacterium tuberculosis H37Rv with an IC50 of 6 nM. DprE1-IN-8 is suitable for research applications focused on tuberculosis and can contribute to the exploration of new therapeutic strategies targeting this pathogen.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	2679830-77-2
Applications	DprE1 Inhibitor
Formula	C₁₉H₁₂F₃N₅O₄S
Molecular Weight	463.39
SMILES	CN(C1=NC(C2=CC(C(F)(F)F)=CC([N+]([O-])=O)=C2S1)=O)CC3=NN=C(O3)C4=CC=CC=C4

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.