EPZ004777 hydrochloride

Catalog No.: A21766

DOT1L inhibitor

EPZ004777 hydrochloride

EPZ004777 hydrochloride Chemical Structure

CAS NO. 1380316-03-9

EPZ004777 hydrochloride is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.

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Biological Activity

EPZ004777 hydrochloride is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.36 mL 86.79 mL 173.57 mL
0.5 mM 3.47 mL 17.36 mL 34.71 mL
1 mM 1.74 mL 8.68 mL 17.36 mL
5 mM 0.35 mL 1.74 mL 3.47 mL

*The above data is based on the productmolecular weight 576.13. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21766
Actions Inhibitor
CAS No. 1380316-03-9
Formula C28H42ClN7O4
M. Wt 576.13
Purity >98%
Synonyms EPZ 004777, EPZ-004777
SMILES NC1=C2C(N([[email protected]]3[[email protected]](O)[[email protected]](O)[[email protected]@H](CN(C(C)C)CCCNC(NC4=CC=C(C(C)(C)C)C=C4)=O)O3)C=C2)=NC=N1.[H]Cl

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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