GPBAR1-IN-3

Catalog No.: A60403
GPBAR1 Agonist/CysLT1R Antagonist
GPBAR1-IN-3 is a selective agonist for the G protein-coupled receptor GPBAR1, exhibiting an EC50 of 0.17 μM. Additionally, it functions as an antagonist of the CysLT1 receptor. This compound is valuable for research into inflammatory processes and potential therapeutic strategies involving GPBAR1 activation and CysLT1R inhibition in various biological contexts.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionGPBAR1-IN-3 is a selective agonist for the G protein-coupled receptor GPBAR1, exhibiting an EC50 of 0.17 μM. Additionally, it functions as an antagonist of the CysLT1 receptor. This compound is valuable for research into inflammatory processes and potential therapeutic strategies involving GPBAR1 activation and CysLT1R inhibition in various biological contexts.
Product Information
Catalog NumA60403
FormulaC21H23NO2
Molecular Weight321.41
CAS Number2760546-05-0
SMILESCC(CC)COC1=CC(OCC2=NC3=C(C=C2)C=CC=C3)=CC=C1
Useful Calculator

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