Linagliptin-d3-1

Catalog No.: A26872
Isotope-Labeled Compounds
Linagliptin-d3-1 is a deuterium-labeled analog of Linagliptin, a highly potent and selective inhibitor of dipeptidyl peptidase-4 (DPP-4) with an IC50 of 1 nM. This isotope-labeled compound is primarily utilized in pharmacokinetic studies and metabolic research to trace the pharmacological pathways of DPP-4 inhibitors in various biological systems. Its unique isotopic signature allows for enhanced detection and quantification in analytical applications, facilitating insights into drug metabolism and efficacy.
Grouped product items
Size Price Stock Qty
1mg
$650.00
In stock
5mg
$2,010.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionLinagliptin-d3-1 is a deuterium-labeled analog of Linagliptin, a highly potent and selective inhibitor of dipeptidyl peptidase-4 (DPP-4) with an IC50 of 1 nM. This isotope-labeled compound is primarily utilized in pharmacokinetic studies and metabolic research to trace the pharmacological pathways of DPP-4 inhibitors in various biological systems. Its unique isotopic signature allows for enhanced detection and quantification in analytical applications, facilitating insights into drug metabolism and efficacy.
Product Information
Catalog NumA26872
FormulaC25H25D3N8O2
Molecular Weight475.56
CAS Number1398044-48-8
SMILESO=C1N(C2=C(C(N1CC3=NC(C)=C4C=CC=CC4=N3)=O)N(CC#CC([2H])([2H])[2H])C(N5CCC[C@@H](N)C5)=N2)C
SynonymsBI 1356-d3-1
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2