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(-)-MK 801 maleate

Catalog No.: A13435

NMDA receptor antagonist.

(-)-MK 801 maleate

(-)-MK 801 maleate Chemical Structure

CAS NO. 121917-57-5

(-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel.

Availability: In stock

Package Price Qty
25 mg
$100.00
50 mg
$185.00
100 mg
$320.00
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Biological Activity

(-)-MK 801 maleate acts as a potent, selective, and non-competitive NMDA receptor antagonist. It acts by binding to a site located within the NMDA associated ion channel.
Targets
NMDA Receptor
30.5 nM(Ki)
In vitro (25°C) DMSO 63 mg/mL (186.73 mM)
Water Insoluble
Ethanol 7 mg/mL (20.74 mM)
In vivo 2% DMSO+40% PEG 300+2% Tween 80+ddH2O 7 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.64 mL 148.21 mL 296.41 mL
0.5 mM 5.93 mL 29.64 mL 59.28 mL
1 mM 2.96 mL 14.82 mL 29.64 mL
5 mM 0.59 mL 2.96 mL 5.93 mL

*The above data is based on the productmolecular weight 337.37. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13435
Actions Antagonist
CAS No. 121917-57-5
Formula C20H19NO4
M. Wt 337.37
Purity >98%
Synonyms MK801, MK-801
SMILES C[C@]12C3=CC=CC=C3C[C@H](N1)C4=CC=CC=C24.C(=C/C(=O)O)\C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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