Opiranserin is a dual antagonist of the glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), exhibiting IC50 values of 0.86 μM and 1.3 μM, respectively. Additionally, it demonstrates antagonistic activity on the recombinant P2X3 receptor with an IC50 of 0.87 μM. This compound is being developed as an injectable analgesic for the management of postoperative pain, highlighting its potential utility in pain research and pharmacological studies.
Opiranserin is a dual antagonist of the glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), exhibiting IC50 values of 0.86 μM and 1.3 μM, respectively. Additionally, it demonstrates antagonistic activity on the recombinant P2X3 receptor with an IC50 of 0.87 μM. This compound is being developed as an injectable analgesic for the management of postoperative pain, highlighting its potential utility in pain research and pharmacological studies.
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