PBRM1-BD2-IN-1 is a selective inhibitor targeting the bromodomain of PBRM1, exhibiting significant binding affinity with a Kd of 0.7 μM and an IC50 of 0.2 μM. This compound demonstrates potent inhibitory activity, making it a valuable tool for probing the role of PBRM1 in cancer biology. PBRM1-BD2-IN-1 is suitable for research applications focused on cancer mechanisms and the therapeutic potential of bromodomain inhibition.
PBRM1-BD2-IN-1 is a selective inhibitor targeting the bromodomain of PBRM1, exhibiting significant binding affinity with a Kd of 0.7 μM and an IC50 of 0.2 μM. This compound demonstrates potent inhibitory activity, making it a valuable tool for probing the role of PBRM1 in cancer biology. PBRM1-BD2-IN-1 is suitable for research applications focused on cancer mechanisms and the therapeutic potential of bromodomain inhibition.
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