PBRM1-BD2-IN-4 is a selective inhibitor of the PBRM1 bromodomain, exhibiting Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, with an IC50 of 0.2 μM for PBRM1-BD2. This compound is instrumental in studying the role of PBRM1 in cancer biology and may contribute to the development of anticancer therapies targeting bromodomain-containing proteins. Its high potency and specificity make it a valuable tool for research focused on epigenetic regulation in cancer contexts.
PBRM1-BD2-IN-4 is a selective inhibitor of the PBRM1 bromodomain, exhibiting Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, with an IC50 of 0.2 μM for PBRM1-BD2. This compound is instrumental in studying the role of PBRM1 in cancer biology and may contribute to the development of anticancer therapies targeting bromodomain-containing proteins. Its high potency and specificity make it a valuable tool for research focused on epigenetic regulation in cancer contexts.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
