PBRM1-BD2-IN-8

Name: PBRM1-BD2-IN-8
Brand: Adooq Bioscience
SKU: A24382
Rating: 5 (288 reviews)

Catalog No.: A24382

PBRM1 Bromodomain inhibitor

PBRM1-BD2-IN-8 (compound 34) is a potent inhibitor of the PBRM1 bromodomain, with a Kd of 4.4 μM and an IC50 of 0.16 μM for PBRM1-BD2, and a Kd of 25 μM for PBRM1-BD5. It exhibits anti-cancer activity.

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PBRM1-BD2-IN-8 2819989-75-6 PBRM1 Bromodomain inhibitor

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Grouped product items
Size	Price	Stock
1mg	$162.00	In stock
5mg	$486.00	In stock
10mg	$828.00	In stock
50mg	$2,484.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description	PBRM1-BD2-IN-8 (compound 34) is a potent inhibitor of the PBRM1 bromodomain, with a Kd of 4.4 μM and an IC50 of 0.16 μM for PBRM1-BD2, and a Kd of 25 μM for PBRM1-BD5. It exhibits anti-cancer activity.

Product Information

Catalog Num	A24382
Formula	C15H13BrN2O
Molecular Weight	317.18
CAS Number	2819989-75-6
SMILES	O=C1NC(C2=CC=CC(C)=C2)NC3=C1C(Br)=CC=C3
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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