Biological Activity
PF-04971729 is a potent and selective inhibitor of the sodium-dependent glucose cotransporter 2.
In vitro | DMSO | 86 mg/mL (196.84 mM) | |
Water | 86 mg/mL (196.84 mM) | ||
Ethanol | 86 mg/mL (196.84 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 22.89 mL | 114.44 mL | 228.89 mL |
0.5 mM | 4.58 mL | 22.89 mL | 45.78 mL |
1 mM | 2.29 mL | 11.44 mL | 22.89 mL |
5 mM | 0.46 mL | 2.29 mL | 4.58 mL |
*The above data is based on the productmolecular weight 436.9 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A11102 |
---|---|
Actions | Inhibitor |
CAS No. | 1210344-57-2 |
Formula | C22H25ClO7 |
M. Wt | 436.9 |
Purity | >98% |
Synonyms | PF04971729, PF 04971729 |
SMILES | CCOC1=CC=C(C=C1)CC2=C(C=CC(=C2)[[email protected]@]34[[email protected]@H]([[email protected]]([[email protected]@H]([[email protected]@](O3)(CO4)CO)O)O)O)Cl |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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