(Rac)-Nebivolol-d4 hydrochloride

Catalog No.: A58826
Stable Isotope
(Rac)-Nebivolol-d4 hydrochloride is a stable isotope-labeled analog of racemic Nebivolol, which serves as a selective β1-adrenergic receptor inhibitor with an IC50 of 0.8 nM. This reagent is primarily utilized in pharmacokinetic studies and metabolic profiling, offering insights into drug metabolism and receptor interactions in various biological systems. Its application in research facilitates a deeper understanding of adrenergic signaling pathways and cardiovascular pharmacotherapy.
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Size Price Stock Qty
1mg
$315.00
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Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Biological Activity
Description(Rac)-Nebivolol-d4 hydrochloride is a stable isotope-labeled analog of racemic Nebivolol, which serves as a selective β1-adrenergic receptor inhibitor with an IC50 of 0.8 nM. This reagent is primarily utilized in pharmacokinetic studies and metabolic profiling, offering insights into drug metabolism and receptor interactions in various biological systems. Its application in research facilitates a deeper understanding of adrenergic signaling pathways and cardiovascular pharmacotherapy.
Product Information
Catalog NumA58826
FormulaC22H22D4ClF2NO4
Molecular Weight445.92
CAS Number2701283-32-9
SMILES[2H]C(NC([2H])(C(C1CCC2=C(O1)C=CC(F)=C2)O)[2H])(C(C3CCC4=CC(F)=CC=C4O3)O)[2H].Cl
Synonyms(Rac)-R 065824-d4 hydrochloride
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