PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 uM for μ-Calpain, about 20-fold selectivity over m-calpain.
Targets
Target
Value
Product Information
Catalog Num
A14245
Formula
C11H8FNO2S
Molecular Weight
237.25
CAS Number
179461-52-0
SMILES
C1=CC2=C(C=C1F)C(=CN2)/C=C(/C(=O)O)\S
Synonyms
PD-151746,PD151746
Storage
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
Solubility
In vitro
DMSO
40 mg/mL (168.6 mM)
Water
Insoluble
Ethanol
40 mg/mL (168.6 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula: