SB 243213 hydrochloride is a selective antagonist of the 5-HT2C receptor with high affinity, exhibiting a pKi of 9.37 and a pKb of 9.8 for the human receptor. This compound demonstrates over 100-fold selectivity for the 5-HT2C receptor compared to various neurotransmitter receptors, enzymes, and ion channels. Its anxiolytic properties indicate potential applications in research related to schizophrenia and motor disorders.
SB 243213 hydrochloride is a selective antagonist of the 5-HT2C receptor with high affinity, exhibiting a pKi of 9.37 and a pKb of 9.8 for the human receptor. This compound demonstrates over 100-fold selectivity for the 5-HT2C receptor compared to various neurotransmitter receptors, enzymes, and ion channels. Its anxiolytic properties indicate potential applications in research related to schizophrenia and motor disorders.
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