SB 243213 is a selective and high-affinity antagonist of the 5-HT2C receptor, exhibiting a pKi of 9.37 and a pKb of 9.8 for the human receptor. This compound demonstrates over 100-fold selectivity against a variety of neurotransmitter receptors, enzymes, and ion channels. SB 243213 shows an improved anxiolytic profile, making it a potential candidate for research applications related to schizophrenia and motor disorders.
SB 243213 is a selective and high-affinity antagonist of the 5-HT2C receptor, exhibiting a pKi of 9.37 and a pKb of 9.8 for the human receptor. This compound demonstrates over 100-fold selectivity against a variety of neurotransmitter receptors, enzymes, and ion channels. SB 243213 shows an improved anxiolytic profile, making it a potential candidate for research applications related to schizophrenia and motor disorders.
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