Talarozole
CYP26 inhibitor/RAMBA
Important Notice: For research use only. We do not sell to patients.
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CYP26 inhibitor/RAMBA
Important Notice: For research use only. We do not sell to patients.
Not your Region? View all Distributors
Discription | Talarozole (R115866) is an oral systemic all-trans retinoic acid metabolism blocking agent (RAMBA) which increases intracellular levels of endogenous all-trans retinoic acid (RA). Talarozole inhibits both CYP26A1 and CYP26B1 with IC50s of 5.4 and 0.46 nM, respectively. | ||
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Catalog Num | A21124 |
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Formula | C21H23N5S |
Molecular Weight | 377.51 |
CAS Number | 201410-53-9 |
SMILES | CCC(CC)C(C1=CC=C(NC2=NC3=CC=CC=C3S2)C=C1)N4N=CN=C4 |
Synonyms | R115866, R 115866, R-115866 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2