Tasimelteon-d5

Catalog No.: A61734
Stable Isotope
Tasimelteon-d5 is a deuterium-labeled derivative of Tasimelteon, a selective dual melatonin receptor agonist targeting MT1 and MT2 receptors. This compound exhibits significantly higher affinity for the MT2 receptor, with an affinity range of 2.1-4.4 times greater than that for the MT1 receptor. Tasimelteon serves as a circadian regulator and is being investigated for its potential therapeutic applications in managing Non-24-Hour Sleep-Wake Disorder (Non-24).
Grouped product items
Size Price Stock Qty
1mg
$415.00
In stock
5mg
$3,225.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionTasimelteon-d5 is a deuterium-labeled derivative of Tasimelteon, a selective dual melatonin receptor agonist targeting MT1 and MT2 receptors. This compound exhibits significantly higher affinity for the MT2 receptor, with an affinity range of 2.1-4.4 times greater than that for the MT1 receptor. Tasimelteon serves as a circadian regulator and is being investigated for its potential therapeutic applications in managing Non-24-Hour Sleep-Wake Disorder (Non-24).
Product Information
Catalog NumA61734
FormulaC15H14D5NO2
Molecular Weight250.35
CAS Number1962124-51-1
SMILES[H][C@]1(C[C@H]1CNC(C([2H])(C([2H])([2H])[2H])[2H])=O)C2=C3CCOC3=CC=C2
SynonymsBMS-214778-d5; VEC-162-d5
Useful Calculator

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