Melatonin Receptors

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  1. MT1/MT2 agonist

    Melatonin is a endogenous hormone that acts as an agonist at melatonin receptors MT1 and MT2.
  2. MT1/MT2-Receptor Agonist

    Ramelteon is a melatonin receptor agonist with both high affinity for melatonin MT1 (IC50 =28.5 ?? 8.55 pM)and MT2 (20.1 ?? 9.25 pM)receptors and selectivity over the MT3 receptor.
  3. Prazosin HCl is an α1 and α2B-adrenoceptor antagonist. Also a potent antagonist at the melatonin MT3 receptor (Ki = 10.2 nM).
  4. MT1 and MT2 receptor agonist

    Tasimelteon is a melatonin MT1 and MT2 receptor agonist.
  5. melanocortin receptor (MR) agonist

    AP1189 is a biased agonist at receptors MC1 and MC3. AP1189 reduced cytokine release, an effect reliant on both MC1 and MC3 as evident from the use of Mc1r(-/-) and Mc3r(-/-) macrophages.
  6. Melatonin receptor agonist

    ACH-000143 is a potent and peripherally preferred melatonin receptor agonist.
  7. MT1/MT2 antagonist

    Luzindole, also known as N-0774, and N-acetyl-2-benzyltryptamine, is a melatonin receptor antagonist that preferentially targets MT1B over MT1A (Ki values are = 10-27 and 158-513 nM, respectively).

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