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Biological Activity
Timegadine, a new antiinflammatory agent, is found to be a potent, competitive inhibitor of cyclo-oxygenase (COX) and lipo-oxygenase, with IC50s ranging from 5 nM (washed rabbit platelets) to 20 μM (rat brain) for COX and 100 μM for lipo-oxygenase both in the cytosol fraction of horse platelet homogenates, and in washed rabbit platelets.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 27.36 mL | 136.8 mL | 273.6 mL |
| 0.5 mM | 5.47 mL | 27.36 mL | 54.72 mL |
| 1 mM | 2.74 mL | 13.68 mL | 27.36 mL |
| 5 mM | 0.55 mL | 2.74 mL | 5.47 mL |
*The above data is based on the productmolecular weight 365.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A17108 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 71079-19-1 |
| Formula | C20H23N5S |
| M. Wt | 365.5 |
| Purity | >98% |
| Synonyms | SR 1368, SR-1368, SR1368 |
| SMILES | CC1=NC2=CC=CC=C2C(/N=C(NC3CCCCC3)/NC4=NC=CS4)=C1 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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