Trelagliptin-13C,d3

Catalog No.: A43545
Stable Isotope
Trelagliptin-13C,d3 is a stable isotope-labeled derivative of Trelagliptin, a highly selective DPP-4 inhibitor with an IC50 value of 4 nM. This compound is utilized in research applications aimed at understanding the pharmacokinetics and pharmacodynamics of glycemic control in type 2 diabetes mellitus (T2DM). Its deuterated form allows for precise tracking in metabolic studies, facilitating deeper insights into the therapeutic effects of DPP-4 inhibition.
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Size Price Stock Qty
1mg
$2,110.00
In stock
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Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Biological Activity
DescriptionTrelagliptin-13C,d3 is a stable isotope-labeled derivative of Trelagliptin, a highly selective DPP-4 inhibitor with an IC50 value of 4 nM. This compound is utilized in research applications aimed at understanding the pharmacokinetics and pharmacodynamics of glycemic control in type 2 diabetes mellitus (T2DM). Its deuterated form allows for precise tracking in metabolic studies, facilitating deeper insights into the therapeutic effects of DPP-4 inhibition.
Product Information
Catalog NumA43545
FormulaC1713CH17D3FN5O2
Molecular Weight361.39
CAS Number2707203-34-5
SMILESN#CC1=CC=C(F)C=C1CN(C(N2[13C]([2H])([2H])[2H])=O)C(N3C[C@H](N)CCC3)=CC2=O
SynonymsSYR-472-13C,d3
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