AG-1024 (Tyrphostin)

AG-1024 (Tyrphostin) is a specific inhibitor of insulin-like growth factor-1 (IGF-1) and insulin receptor tyrosine kinase activity. Exhibits lower IC50 values for IGF-1 than for the insulin receptor. Also inhibits insulin-stimulated cellular proliferation.
Grouped product items
Product Name Price Stock Qty
AG-1024 (Tyrphostin) 5mg
$60.00
In stock
AG-1024 (Tyrphostin) 10mg
$110.00
In stock
AG-1024 (Tyrphostin) 25mg
$220.00
In stock
AG-1024 (Tyrphostin) 50mg
$350.00
In stock
AG-1024 (Tyrphostin) 10mM * 1mL in DMSO
$70.00
In stock
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Adooq Products cited in reputable paper
Adooq's AG-1024 (Tyrphostin) has been cited by 1 publications
  • Maeda A, .et al. , Mol Nutr Food Res. , 2014, 58(6):1177-89 PMID: 24668740
  • Biological Activity
    Discription AG-1024 (Tyrphostin) is a specific inhibitor of insulin-like growth factor-1 (IGF-1) and insulin receptor tyrosine kinase activity. Exhibits lower IC50 values for IGF-1 than for the insulin receptor. Also inhibits insulin-stimulated cellular proliferation.
    Targets
    Target Value
    Product Information
    Catalog Num A11400
    Formula C14H13BrN2O
    Molecular Weight 305.2
    CAS Number 65678-07-1
    SMILES CC(C)(C)C1=C(C(=CC(=C1)C=C(C#N)C#N)Br)O
    Synonyms AG1024
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro (25°C) DMSO 59 mg/mL (193.33 mM)
    Water Insoluble
    Ethanol Insoluble
    In vivo 1% DMSO+30% polyethylene glycol+1% Tween 80 28 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 32.77 mL 163.83 mL 327.65 mL
    0.5 mM 6.55 mL 32.77 mL 65.53 mL
    1 mM 3.28 mL 16.38 mL 32.77 mL
    5 mM 0.66 mL 3.28 mL 6.55 mL
    Useful Calculator

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    This equation is commonly abbreviated as: C1V1 = C2V2

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