Imatinib Mesylate

ON SALE

Bcr-Abl inhibitor

0 Customer Reviews
Catalog No. A10468

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Imatinib Mesylate 100mg A10468-100

Regular Price: $60.00

Special Price: $51.00

Imatinib Mesylate 200mg A10468-200

Regular Price: $100.00

Special Price: $85.00

Imatinib Mesylate 500mg A10468-500

Regular Price: $160.00

Special Price: $136.00

Imatinib Mesylate 10mM * 1mL in DMSO A10468-10mM-D

Regular Price: $63.00

Special Price: $53.55

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Imatinib mesylate, a selective tyrosine kinase inhibitor, induced a sustained objective response in treating gastrointestinal stromal tumors with the inhibition of the KIT signal-transduction pathway.

Imatinib Mesylate

Double click on above image to view full picture

Zoom Out
Zoom In

More Views

Publications citing Adooq Products

Chemical Information

Catalog Num A10468
Actions Inhibitor
M. Wt 589.7
Formula C29H31N7O.CH4SO3
Solubility DMSO
Purity >98%
Storage at -20°C 2 years
CAS No. 220127-57-1
Synonyms Gleevec, Glivec, CGP-57148B, STI-571
SMILES code CC1=C(C=C(C=C1)NC(=O)C2=CC=C(C=C2)CN3CCN(CC3)C)NC4=NC=CC(=N4)C5=CN=CC=C5.CS(=O)(=O)O
Chemical Name 4-(4-Methylpiperazin-1-ylmethyl)-N-[4-methyl-3-[4-(3-pyridyl)pyrimidin-2-ylamino]phenyl]benzamide methanesulfonate

Biological Activity

Description
Imatinib mesylate, a selective tyrosine kinase inhibitor, induced a sustained objective response in treating gastrointestinal stromal tumors with the inhibition of the KIT signal-transduction pathway.
Targets
PDGFR (Cell-free assay) c-Kit (M-07e cells) v-Abl (Cell-free assay)
100 nM100 nM600 nM

Solubility

Solubility (25°C) * In vitro DMSO 118 mg/mL (200.09 mM)
Water 118 mg/mL (200.09 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo Saline 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

View Related Products By Research Topics

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.


Keywords:buy Imatinib Mesylate | Imatinib Mesylate Supplier | purchase Imatinib Mesylate | Imatinib Mesylate cost | Imatinib Mesylate manufacturer | order Imatinib Mesylate | Imatinib Mesylate distributor | buy 220127-57-1| 220127-57-1 Supplier | purchase 220127-57-1 | 220127-57-1 cost | 220127-57-1 manufacturer | order 220127-57-1 | 220127-57-1 distributor