A 922500

Catalog No.: A11199

DGAT-1 inhibitor

A 922500

A 922500 Chemical Structure

CAS NO. 959122-11-3

A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
50 mg
$400.00
100 mg
$700.00
10mM * 1mL in DMSO
$128.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).

Targets
human DGAT-1 mouse DGAT-1 DGAT-2
7 nM24 nM53 μM
In vitro (25°C) DMSO 86 mg/mL (200.7 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 15% Captisol 20 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.34 mL 116.69 mL 233.38 mL
0.5 mM 4.67 mL 23.34 mL 46.68 mL
1 mM 2.33 mL 11.67 mL 23.34 mL
5 mM 0.47 mL 2.33 mL 4.67 mL

*The above data is based on the productmolecular weight 428.48. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11199
Actions Inhibitor
M. Wt 428.48
Formula C26H24N2O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 959122-11-3
Synonyms DGAT-1 Inhibitor 4a, A-922500, A922500
SMILES C1C[[email protected]]([[email protected]@H](C1)C(=O)O)C(=O)C2=CC=C(C=C2)C3=CC=C(C=C3)NC(=O)NC4=CC=CC=C4

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy A 922500 | A 922500 Supplier | purchase A 922500 | A 922500 cost | A 922500 manufacturer | order A 922500 | A 922500 distributor | buy 959122-11-3| 959122-11-3 Supplier | purchase 959122-11-3 | 959122-11-3 cost | 959122-11-3 manufacturer | order 959122-11-3 | 959122-11-3 distributor
Rewards