A 922500
A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).
Important Notice: For research use only. We do not sell to patients.
A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively).
Important Notice: For research use only. We do not sell to patients.
Discription | A 922500 is a diacylglycerol acyltransferase 1 (DGAT-1) inhibitor (IC50 values are 7 and 24 nM at human and mouse DGAT-1 respectively). |
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Catalog Num | A11199 |
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Formula | C26H24N2O4 |
Molecular Weight | 428.48 |
CAS Number | 959122-11-3 |
SMILES | C1C[C@H]([C@@H](C1)C(=O)O)C(=O)C2=CC=C(C=C2)C3=CC=C(C=C3)NC(=O)NC4=CC=CC=C4 |
Synonyms | DGAT-1 Inhibitor 4a, A-922500, A922500 |
Storage | Store lyophilized at -20ºC, keep desiccated. |
In vitro (25°C) | DMSO | 83 mg/mL (193.7 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 15% Captisol | 19 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 23.34 mL | 116.69 mL | 233.38 mL |
0.5 mM | 4.67 mL | 23.34 mL | 46.68 mL |
1 mM | 2.33 mL | 11.67 mL | 23.34 mL |
5 mM | 0.47 mL | 2.33 mL | 4.67 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2