BRD4-IN-10

Catalog No.: A40450
BRD4 Inhibitor
BRD4-IN-10 is a selective inhibitor of Bromodomain-containing protein 4 (BRD4), exhibiting an IC50 of 13.5 nM. This compound demonstrates anti-inflammatory and anti-fibrotic activities, making it a valuable tool in studies related to renal fibrosis. It also possesses favorable metabolic stability and pharmacokinetic properties, enhancing its suitability for research applications in exploring BRD4-related pathways and therapeutic interventions.
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50mg
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Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Nature Volume 622 Issue 7982 (2023)
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Nature volume 551, pages639-643 (2017)
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Biological Activity
DescriptionBRD4-IN-10 is a selective inhibitor of Bromodomain-containing protein 4 (BRD4), exhibiting an IC50 of 13.5 nM. This compound demonstrates anti-inflammatory and anti-fibrotic activities, making it a valuable tool in studies related to renal fibrosis. It also possesses favorable metabolic stability and pharmacokinetic properties, enhancing its suitability for research applications in exploring BRD4-related pathways and therapeutic interventions.
Product Information
Catalog NumA40450
FormulaC24H30N8O3
Molecular Weight478.55
CAS Number3051852-76-4
SMILESO=C1NC(C2(CCN(C3=NC(NC4=CC(N(C(C)C)[C@H](C)C(N5C)=O)=C5C=C4)=NC=C3)CC2)N1)=O
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