GNE-272

Catalog No.: A12474

GNE-272

GNE-272 Chemical Structure

CAS NO. 1936428-93-1

GNE-272 is a potent and selective in vivo probe for the bromodomains of CBP/EP300 with IC50 values of 0.02, 0.03 and 13 μM for CBP, EP300 and BRD4, respectively.

Availability: In stock

Package Price Qty
2 mg
$119.00
5 mg
$238.00
10 mg
$357.00
50 mg
$2,380.00
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Biological Activity

GNE-272 is a potent and selective in vivo probe for the bromodomains of CBP/EP300 with IC50 values of 0.02, 0.03 and 13 μM for CBP, EP300 and BRD4, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.56 mL 117.79 mL 235.59 mL
0.5 mM 4.71 mL 23.56 mL 47.12 mL
1 mM 2.36 mL 11.78 mL 23.56 mL
5 mM 0.47 mL 2.36 mL 4.71 mL

*The above data is based on the productmolecular weight 424.47. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12474
CAS No. 1936428-93-1
Formula C22H25FN6O2
M. Wt 424.47
Purity >98%
Synonyms GNE 272, GNE272
SMILES CC(N1CCC2=C(C(NC3=C(F)C=C(C4=CN(C)N=C4)C=C3)=NN2[[email protected]@H]5COCC5)C1)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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