PFI-1
PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4.
Free Delivery on orders over $500
Research use only. We do not sell to patients.
Loading distributor info...
Adooq Products cited in reputable paper
Adooq's PFI-1 has been cited by 1 publications
- Lisa-Maria Winter, .et al. , Sci Rep, 2023, Jul 26;13(1):12061 PMID: 37495707
Biological Activity
| Description | PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4. | |||||
|---|---|---|---|---|---|---|
| Targets |
| |||||
| Cell Research |
|
Product Information
| Catalog Num | A12545 |
|---|---|
| Formula | C16H17N3O4S |
| Molecular Weight | 347.39 |
| CAS Number | 1403764-72-6 |
| SMILES | CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O |
| Synonyms | PFI 1, PFI1 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
Solubility
| In vitro | DMSO | 65 mg/mL (187.11 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| * <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. | |||
Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 28.79 mL | 143.93 mL | 287.86 mL |
| 0.5 mM | 5.76 mL | 28.79 mL | 57.57 mL |
| 1 mM | 2.88 mL | 14.39 mL | 28.79 mL |
| 5 mM | 0.58 mL | 2.88 mL | 5.76 mL |
Useful Calculator
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)
Please check COA/MSDS for correct molecular weight.
Calculate the dilution required to prepare a stock solution.This equation is commonly abbreviated as: C1V1 = C2V2
