PFI-1

Name: PFI-1
SKU: A12545
Price: 50 USD
Rating: 5 (1 reviews)

Catalog No.: A12545

BET inhibitor

Adooq's PFI-1 has been cited by 1 publications

PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4.

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

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Adooq Products cited in reputable paper

Adooq's PFI-1 has been cited by 1 publications

Lisa-Maria Winter, .et al. , Sci Rep, 2023, Jul 26;13(1):12061 PMID: 37495707

Biological Activity

Discription

PFI-1 is a BET bromodomain inhibitor that exhibits inhibitory activity at BRD2 and BRD4.

Targets

Target	Value

Chemical Information

Catalog Num	A12545
Formula	C16H17N3O4S
Molecular Weight	347.39
CAS Number	1403764-72-6
SMILES	CN1CC2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O
Synonyms	PFI 1, PFI1
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro	DMSO	65 mg/mL (187.11 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	28.79 mL	143.93 mL	287.86 mL
0.5 mM	5.76 mL	28.79 mL	57.57 mL
1 mM	2.88 mL	14.39 mL	28.79 mL
5 mM	0.58 mL	2.88 mL	5.76 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Product Name	Price	Stock
PFI-1 5mg	$50.00	In stock
PFI-1 10mg	$80.00	In stock
PFI-1 25mg	$150.00	In stock
PFI-1 50mg	$220.00	In stock
*PFI-1 10mM 1mL in DMSO**	$94.00	In stock