I-BET787 is an orally active inhibitor of bromodomain and extraterminal (BET) proteins, specifically targeting BRD4 with pIC50 values of 7.1 for BD1 and 5.9 for BD2. This compound exhibits anti-inflammatory properties in murine models, making it a valuable tool for studying inflammatory pathways and the role of BET proteins in various diseases. I-BET787 is utilized in research focused on cancer, cardiovascular diseases, and autoimmune disorders.
I-BET787 is an orally active inhibitor of bromodomain and extraterminal (BET) proteins, specifically targeting BRD4 with pIC50 values of 7.1 for BD1 and 5.9 for BD2. This compound exhibits anti-inflammatory properties in murine models, making it a valuable tool for studying inflammatory pathways and the role of BET proteins in various diseases. I-BET787 is utilized in research focused on cancer, cardiovascular diseases, and autoimmune disorders.
This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:
