Pelanserin is an orally active antihypertensive agent that primarily functions as a potent 5-HT2 receptor antagonist. It effectively inhibits α-adrenergic receptor activity, showcasing an ED50 value of 0.03 μg/mL. Additionally, Pelanserin demonstrates vasodilatory properties with an ED100 of 5 μg. This compound is valuable for research applications focused on hypertension, proving effective in hypertensive rodent models and renal hypertensive dog breeds.
Pelanserin is an orally active antihypertensive agent that primarily functions as a potent 5-HT2 receptor antagonist. It effectively inhibits α-adrenergic receptor activity, showcasing an ED50 value of 0.03 μg/mL. Additionally, Pelanserin demonstrates vasodilatory properties with an ED100 of 5 μg. This compound is valuable for research applications focused on hypertension, proving effective in hypertensive rodent models and renal hypertensive dog breeds.
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