PF-543 Citrate

Catalog No.: A15210

SphK1 Inhibitor

PF-543 Citrate

PF-543 Citrate Chemical Structure

CAS NO. 1415562-83-2

PF-543 Citrate is a novel cell-permeant inhibitor of SphK1 with a K(i) of 3.6 nM, PF-543 is sphingosine-competitive and is more than 100-fold selective for SphK1 over the SphK2 isoform.

Availability: In stock

Package Price Qty
5 mg
$110.00
10 mg
$190.00
50 mg
$700.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PF-543 Citrate is a novel cell-permeant inhibitor of SphK1 with a K(i) of 3.6 nM, PF-543 is sphingosine-competitive and is more than 100-fold selective for SphK1 over the SphK2 isoform.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.2 mL 76.02 mL 152.04 mL
0.5 mM 3.04 mL 15.2 mL 30.41 mL
1 mM 1.52 mL 7.6 mL 15.2 mL
5 mM 0.3 mL 1.52 mL 3.04 mL

*The above data is based on the productmolecular weight 657.73. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A15210
Actions Inhibitor
M. Wt 657.73
Formula C33H39NO11S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1415562-83-2
Synonyms PF543 Citrate, PF 543 Citrate
SMILES CC1=CC(=CC(=C1)OCC2=CC=C(C=C2)CN3CCCC3CO)CS(=O)(=O)C4=CC=CC=C4.C(C(=O)O)C(CC(=O)O)(C(=O)O)O

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy PF-543 Citrate | PF-543 Citrate Supplier | purchase PF-543 Citrate | PF-543 Citrate cost | PF-543 Citrate manufacturer | order PF-543 Citrate | PF-543 Citrate distributor | buy 1415562-83-2| 1415562-83-2 Supplier | purchase 1415562-83-2 | 1415562-83-2 cost | 1415562-83-2 manufacturer | order 1415562-83-2 | 1415562-83-2 distributor
Rewards