CEP-18770 (Delanzomib)

Catalog No.: A11145

Proteasome inhibitor

CEP-18770 (Delanzomib) Chemical Structure

CAS NO. 847499-27-8

CEP-18770 is a novel orally active proteasome inhibitor with a favorable tumor selectivity profile for the treatment of MM and other malignancies responsive to proteasome inhibition.

Availability: In stock Shipped in 7-10 Days

Package Price Qty
5 mg
$70.00
10 mg
$120.00
50 mg
$350.00
100 mg
$600.00
10mM * 1mL in DMSO
$117.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

CEP-18770 is a novel orally active proteasome inhibitor with a favorable tumor selectivity profile for the treatment of MM and other malignancies responsive to proteasome inhibition.
Targets
Chymotrypsin-like proteasome
3.8 nM
In vitro DMSO 83 mg/mL (200.83 mM)
Water <1 mg/mL (<1 mM)
Ethanol 83 mg/mL (200.83 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.2 mL 120.98 mL 241.95 mL
0.5 mM 4.84 mL 24.2 mL 48.39 mL
1 mM 2.42 mL 12.1 mL 24.2 mL
5 mM 0.48 mL 2.42 mL 4.84 mL

*The above data is based on the productmolecular weight 413.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11145
Actions Inhibitor
M. Wt 413.3
Formula C21H28BN3O5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 847499-27-8
Synonyms CEP18770
SMILES B([[email protected]](CC(C)C)NC(=O)[[email protected]]([[email protected]@H](C)O)NC(=O)C1=CC=CC(=N1)C2=CC=CC=C2)(O)O

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