MLN9708

Catalog No.: A10602

Proteasome Inhibitor

MLN9708

MLN9708 Chemical Structure

CAS NO. 1201902-80-8

MLN9708 is a proteasome inhibitor, which inhibits the activity of the proteasome, blocking the targeted proteolysis normally performed by the proteasome.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $60.00

Special Price $54.00

10 mg

Regular Price: $80.00

Special Price $72.00

50 mg

Regular Price: $150.00

Special Price $135.00

100 mg

Regular Price: $250.00

Special Price $225.00

10mM * 1mL in DMSO

Regular Price: $60.00

Special Price $54.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MLN9708 is a proteasome inhibitor, which inhibits the activity of the proteasome, blocking the targeted proteolysis normally performed by the proteasome.
Targets
20S proteasome (Cell-free assay) 20S proteasome (Cell-free assay)
0.93 nM(Ki)3.4 nM
In vitro (25°C) DMSO 100 mg/mL (193.37 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 0.5% hydroxyethyl cellulose 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.34 mL 96.69 mL 193.39 mL
0.5 mM 3.87 mL 19.34 mL 38.68 mL
1 mM 1.93 mL 9.67 mL 19.34 mL
5 mM 0.39 mL 1.93 mL 3.87 mL

*The above data is based on the productmolecular weight 517.1 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A10602
Actions Inhibitor
M. Wt 517.1
Formula C20H23BCl2N2O9
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1201902-80-8
Synonyms MLN-9708
SMILES B1(OC(=O)CC(O1)(CC(=O)O)C(=O)O)[[email protected]](CC(C)C)NC(=O)CNC(=O)C2=C(C=CC(=C2)Cl)Cl

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