MLN9708

Catalog No.: A10602

Proteasome Inhibitor

MLN9708

MLN9708 Chemical Structure

CAS NO. 1201902-80-8

MLN9708 is a proteasome inhibitor, which inhibits the activity of the proteasome, blocking the targeted proteolysis normally performed by the proteasome.

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$80.00
50 mg
$150.00
100 mg
$250.00
10mM * 1mL in DMSO
$60.00
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Biological Activity

MLN9708 is a proteasome inhibitor, which inhibits the activity of the proteasome, blocking the targeted proteolysis normally performed by the proteasome.
Targets
20S proteasome (Cell-free assay) 20S proteasome (Cell-free assay)
0.93 nM(Ki)3.4 nM
In vitro (25°C) DMSO 85 mg/mL (164.36 mM)
Water Insoluble
Ethanol Insoluble
In vivo 0.5% hydroxyethyl cellulose 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.34 mL 96.69 mL 193.39 mL
0.5 mM 3.87 mL 19.34 mL 38.68 mL
1 mM 1.93 mL 9.67 mL 19.34 mL
5 mM 0.39 mL 1.93 mL 3.87 mL

*The above data is based on the productmolecular weight 517.1 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10602
Actions Inhibitor
CAS No. 1201902-80-8
Formula C20H23BCl2N2O9
M. Wt 517.1
Purity >98%
Synonyms MLN-9708
SMILES B1(OC(=O)CC(O1)(CC(=O)O)C(=O)O)[[email protected]](CC(C)C)NC(=O)CNC(=O)C2=C(C=CC(=C2)Cl)Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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