D595

Catalog No.: A26591
Histone Methyltransferase
D595 is a phenylethylamine derivative that functions primarily as a histone methyltransferase inhibitor. This compound exhibits significant biological activity by inhibiting the uptake of monoamine neurotransmitters, displaying a high affinity for the dopamine transporter (DAT), serotonin transporter (SERT), and norepinephrine transporter (NET). Structural modifications, particularly alterations in hydroxyl stereochemistry, can influence its binding interactions with these transporters, demonstrating a specific stereoselectivity. D595 is suitable for studies involving neuropharmacology and epigenetic regulation.
Grouped product items
Size Price Stock Qty
25mg
$1,275.00
In stock
50mg
$1,625.00
In stock
100mg
$2,000.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

Loading distributor info...

Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionD595 is a phenylethylamine derivative that functions primarily as a histone methyltransferase inhibitor. This compound exhibits significant biological activity by inhibiting the uptake of monoamine neurotransmitters, displaying a high affinity for the dopamine transporter (DAT), serotonin transporter (SERT), and norepinephrine transporter (NET). Structural modifications, particularly alterations in hydroxyl stereochemistry, can influence its binding interactions with these transporters, demonstrating a specific stereoselectivity. D595 is suitable for studies involving neuropharmacology and epigenetic regulation.
Product Information
Catalog NumA26591
FormulaC25H32Cl2N2O2
Molecular Weight463.44
CAS Number16740-29-7
SMILESN#CC(CCCN(CCC1=CC=C(C(OC)=C1)OC)C)(C(C)C)C2=CC=C(C(Cl)=C2)Cl
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2