KDM2A/7A-IN-1

Name: KDM2A/7A-IN-1
Brand: Adooq Bioscience
SKU: A19724
Rating: 5 (288 reviews)

Catalog No.: A19724

KDM2A/7A inhibitor

KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16?μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases.

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KDM2A/7A-IN-1 2169272-46-0 KDM2A/7A inhibitor

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Grouped product items
Size	Price	Stock
1mg	$265.00	In stock
5mg	$655.00	In stock
10mg	$1,055.00	In stock
25mg	$2,085.00	In stock
50mg	$2,775.00	In stock
100mg	$3,695.00	In stock
Bulk Size	Bulk Discount

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Data Sheet SDS

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Biological Activity

Description	KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16?μM for KDM2A, exhibits 75 fold selevtivity over other JmjC lysine demethylases, and is inactive on methyl transferases, and histone acetyl transferases.

Product Information

Catalog Num	A19724
Formula	C33H38N4O
Molecular Weight	506.68
CAS Number	2169272-46-0
SMILES	CC(N([C@@H](C1=CN=CC(CCCCCCCN2CCCC2)=C1)[C@@]3(C4=CC=CC=C4)C#N)C5=C3C=CC=C5)=O
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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