Other Inhibitors

Cat. No.

A13768

CAS No.

924416-43-3

AdipoRon

AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)

Cat. No.

A10266

CAS No.

485-35-8

Cytisine (Baphitoxine, Sophorine)

Cytisine is a nicotinic acetylcholine receptor agonist, and as a pharmaceutical preparation it is available for the treatment of nicotinism. It is a pyridine-like alkaloid that can be toxic in high doses. Pharmacologically it exhibits similar effects to nicotine due to structural similarity of the two molecules.

Cat. No.

A10918

CAS No.

312753-06-3

Indacaterol

Synonyms: Arcapta; Onbrez

Indacaterol is an ultra-long-acting beta-adrenoceptor agonist.

Cat. No.

A11670

CAS No.

108341-18-0

Noradrenaline bitartrate monohydrate

Synonyms: Levophed

Noradrenaline bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.

Cat. No.

A11761

CAS No.

635701-59-6

Merck SIP Agonist

Cat. No.

A12568

CAS No.

1005491-05-3

Tirasemtiv (CK-2017357)

Synonyms: CK-2017357

Tirasemtiv amplifies skeletal muscle response to nerve activation in humans.

Cat. No.

A12908

CAS No.

1420071-30-2

Bioymifi

Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.

Cat. No.

A13855

CAS No.

447407-36-5

AC-42 hydrochloride

Synonyms: AC 42

AC 42 is an allosteric agonist.

Cat. No.

A13960

CAS No.

259666-71-2

SM-130686

SM-130686 is a potent, orally active growth hormone secretagogue, with around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.

Cat. No.

A14150

CAS No.

1256037-58-7

TRX 818

TRX-818 is a new, potent and multi-targeted anti-cancer agent in numerous human cancer cell lines.

Cat. No.

A15852

CAS No.

220551-92-8

DAA-1106

Synonyms: DAA 110

DAA-1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), as a potent and selective agonist at the peripheral benzodiazepine receptor.

Cat. No.

A17588

CAS No.

1188-38-1

Carglumic Acid

Synonyms: OE312; AJ 266447; AJ-26647; Carglumic Acid.

Carglumic acid (N-Carbamyl-L-glutamic acid), a functional analogue of N-acetylglutamate (NAG) and a carbamoyl phosphate synthetase 1 (CPS1) activator, is used to treat acute and chronic hyperammonemia associated with NAG synthase (NAGS) deficiency.

Cat. No.

A18152

CAS No.

23642-66-2

Benfluorex hydrochloride

Synonyms: Benfluorex HCl; Lipophoral; Mediator; JP 992; EINECS 245-801-8; Mediaxal; Balans

Benfluorex hydrochloride (JP-992 hydrochloride) is a hepatic nuclear factor 4 alpha (HNF4α) activator.

Cat. No.

A19055

CAS No.

421581-52-4

G6PD activator AG1

G6PD activator AG1 is a glucose-6-phosphate dehydrogenase (G6PD) activator with an EC50 of 3 μ, extracted from patent WO2019023264A1, compound AG1.

Cat. No.

A19359

CAS No.

439685-79-7

Pro-xylane

Synonyms: Hydroxypropyl tetrahydropyrantriol

Pro-xylane (Hydroxypropyl tetrahydropyrantriol) is a biologically active C-glycoside in aqueous media, acts as an activator of glycosaminoglycans (GAGs) biosynthesis.

Cat. No.

A19489

CAS No.

81921-35-9

N6-Methyladenosine 5'-monophosphate disodium salt

N6-Methyladenosine 5'-monophosphate disodium salt is an activator of glycogen phosphorylase b, with a Ka value of 22 µM. N6-Methyladenosine 5'-monophosphate disodium salt is a non-competitive rat adenylate kinase II inhibitor.

Cat. No.

A20007

CAS No.

260553-97-7

TM-25659

TM-25659 is a transcriptional co-activator with PDZ-binding motif (TAZ) modulator. Anti-osteoporotic and anti-obesity activities.