Other Inhibitors

Other Inhibitors groups bioactive small molecules whose targets fall outside the pathway categories of this catalogue. The compounds have not yet been assigned to target categories, so the range is broad and uneven. Streptozotocin, a glucosamine-nitrosourea compound used to induce experimental diabetes in rodents, sits beside the O-GlcNAcase inhibitor Thiamet G. Exherin is an N-cadherin antagonist, and AdipoRon is an agonist of adiponectin receptors 1 and 2 (AdipoR1 and AdipoR2). Plant compounds such as the isoflavone daidzein are also included. Despite the category name, not every compound is an inhibitor, as the AdipoRon example shows. Compounds with a well-defined target are usually listed in the matching pathway or target category.

13 Items

  • AdipoRon
    Cat. No.
    A13768

    AdipoRon

    AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)

    5 mg
    $25.00
    10 mg
    $40.00
    All 9 sizes
  • Bilobalide
    Cat. No.
    A10144

    Bilobalide

    Bilobalide, a biologically active terpenic trilactone (terpinoid), derived from geranylgeranyl pyrophosphate (GGPP) is an inducer of cytochrome P450 enzymes CYP3A1 and CYP1A2. May contain properties to stop apoptosis activation of the phosphatidylinositol 3-Kinase pathway in SH-SY5Y cells.

    5 mg
    $20.00
    10 mg
    $30.00
    All 6 sizes
  • Cytisine (Baphitoxine, Sophorine)
    Cat. No.
    A10266

    Cytisine (Baphitoxine, Sophorine)

    Cytisine is a nicotinic acetylcholine receptor agonist, and as a pharmaceutical preparation it is available for the treatment of nicotinism. It is a pyridine-like alkaloid that can be toxic in high doses. Pharmacologically it exhibits similar effects to nicotine due to structural similarity of the two molecules.

    5 mg
    $20.00
    10 mg
    $30.00
    All 8 sizes
  • Indacaterol
    Cat. No.
    A10918

    Indacaterol

    Synonyms: Arcapta; Onbrez

    Indacaterol is an ultra-long-acting beta-adrenoceptor agonist.

    5 mg
    $20.00
    10 mg
    $30.00
    All 7 sizes
  • Bioymifi
    Cat. No.
    A12908

    Bioymifi

    Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.

    1 mg
    $25.00
    2 mg
    $35.00
    All 8 sizes
  • SM-130686
    Cat. No.
    A13960

    SM-130686

    SM-130686 is a potent, orally active growth hormone secretagogue, with around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.

    Out of stock

    All 2 sizes
  • Neuropathiazol
    Cat. No.
    A14058

    Neuropathiazol

    Neuropathiazol is a synthetic small molecule that induces neuronal differentiation of adult hippocampal neural progenitor cells.

    1 mg
    $40.00
    5 mg
    $110.00
    All 7 sizes
  • ISX-9
    Cat. No.
    A15774

    ISX-9

    Synonyms: Isoxazole 9

    ISX-9 is a small molecule inducer of adult neural stem cell differentiation.

    2 mg
    $35.00
    5 mg
    $60.00
    All 8 sizes
  • DAA-1106
    Cat. No.
    A15852

    DAA-1106

    Synonyms: DAA 110

    DAA-1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), as a potent and selective agonist at the peripheral benzodiazepine receptor.

    2 mg
    $20.00
    5 mg
    $35.00
    All 7 sizes
  • N-(beta-Ketocaproyl)-L-hoMoserine lactone
    Cat. No.
    A22261

    N-(beta-Ketocaproyl)-L-hoMoserine lactone

    N-(beta-ketocaproyl)-L-Homoserine lactone (N-(Ketocaproyl)-L-homoserine lactone, N-(β-Ketocaproyl)-L-hoMoserine lactone) is an autoinducer of P. fischeri luciferase and a component of quorum regulatory sensing.

    5 mg
    $20.00
    10 mg
    $35.00
    All 7 sizes

13 Items

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