Other Inhibitors

Cat. No.

A13768

CAS No.

924416-43-3

AdipoRon

AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)

Cat. No.

A10144

CAS No.

33570-04-6

Bilobalide

Bilobalide, a biologically active terpenic trilactone (terpinoid), derived from geranylgeranyl pyrophosphate (GGPP) is an inducer of cytochrome P450 enzymes CYP3A1 and CYP1A2. May contain properties to stop apoptosis activation of the phosphatidylinositol 3-Kinase pathway in SH-SY5Y cells.

Cat. No.

A10266

CAS No.

485-35-8

Cytisine (Baphitoxine, Sophorine)

Cytisine is a nicotinic acetylcholine receptor agonist, and as a pharmaceutical preparation it is available for the treatment of nicotinism. It is a pyridine-like alkaloid that can be toxic in high doses. Pharmacologically it exhibits similar effects to nicotine due to structural similarity of the two molecules.

Cat. No.

A10918

CAS No.

312753-06-3

Indacaterol

Synonyms: Arcapta; Onbrez

Indacaterol is an ultra-long-acting beta-adrenoceptor agonist.

Cat. No.

A11761

CAS No.

635701-59-6

Merck SIP Agonist

Cat. No.

A12455

CAS No.

162704-20-3

UK-157147

UK-157147 is a substrate for UDP-glucuronosyltransferases (UGT1A1) with a Km value of 105 μM.

Cat. No.

A12908

CAS No.

1420071-30-2

Bioymifi

Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.

Cat. No.

A13789

CAS No.

2591-17-5

D-Luciferin

Synonyms: Firefly Luciferin

D-Luciferin is a popular bioluminescent substrate of luciferase in the presence of ATP, used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications.

Cat. No.

A13855

CAS No.

447407-36-5

AC-42 hydrochloride

Synonyms: AC 42

AC 42 is an allosteric agonist.

Cat. No.

A13960

CAS No.

259666-71-2

SM-130686

SM-130686 is a potent, orally active growth hormone secretagogue, with around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.

Cat. No.

A14058

CAS No.

880090-88-0

Neuropathiazol

Neuropathiazol is a synthetic small molecule that induces neuronal differentiation of adult hippocampal neural progenitor cells.

Cat. No.

A15774

CAS No.

832115-62-5

ISX-9

Synonyms: Isoxazole 9

ISX-9 is a small molecule inducer of adult neural stem cell differentiation.

Cat. No.

A15852

CAS No.

220551-92-8

DAA-1106

Synonyms: DAA 110

DAA-1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), as a potent and selective agonist at the peripheral benzodiazepine receptor.

Cat. No.

A15862

CAS No.

21919-05-1

CB1954

Synonyms: Tretazicar

CB1954 is a anticancer prodrug that is converted in the presence of the enzyme NQO2 and co-substrate caricotamide ( EP-0152R) (EP) into a potent cytotoxic bifunctional alkylating agent.It can be activated by NAD(P)H quinone oxidoreductase 2.

Cat. No.

A15897

CAS No.

55779-48-1

Coelenterazine

Synonyms: CLZN

Coelenterazine is a luminescent enzyme substrate, used for monitoring reporter genes in BRET, ELISA and HTS techniques.

Cat. No.

A16019

CAS No.

1160928-63-1

RETF-4NA

RETF-4NA is a chymase substrate peptide that is cleaved more avidly by α2-macroglobulin-bound chymase than the free, unbound form.

Cat. No.

A16384

CAS No.

61-78-9

4-Aminohippuric Acid

Synonyms: p-Aminohippuric acid

4-Aminohippuric acid is a typical substrate of organic anion transport systems.

Cat. No.

A19054

CAS No.

20902-53-8

L-Lysine thioctate

L-Lysine thioctate is a substrate of lipoamidase.

Cat. No.

A19148

CAS No.

122799-38-6

2'-Fluorothymidine

Synonyms: 2'-Deoxy-2'-fluoro-5-Methyluridine

2'-Fluorothymidine (2'-Fluoro-2'-deoxythymidine), a bioisostere of both thymidine (TdR) and methyluridine, is a putative highly selective substrate for thymidine kinase type 2 (TK2).

Cat. No.

A20542

CAS No.

289479-94-3

TN1

TN1 is a potent fetal hemoglobin (HbF) inducer.

Cat. No.

A22261

CAS No.

143537-62-6

N-(beta-Ketocaproyl)-L-hoMoserine lactone

N-(beta-ketocaproyl)-L-Homoserine lactone (N-(Ketocaproyl)-L-homoserine lactone, N-(β-Ketocaproyl)-L-hoMoserine lactone) is an autoinducer of P. fischeri luciferase and a component of quorum regulatory sensing.