Other Inhibitors

Cat. No.

A13768

CAS No.

924416-43-3

AdipoRon

AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM). IC50 value: 1.8/3.1 uM(AdipoR1/2, Kd)

Cat. No.

A10266

CAS No.

485-35-8

Cytisine (Baphitoxine, Sophorine)

Cytisine is a nicotinic acetylcholine receptor agonist, and as a pharmaceutical preparation it is available for the treatment of nicotinism. It is a pyridine-like alkaloid that can be toxic in high doses. Pharmacologically it exhibits similar effects to nicotine due to structural similarity of the two molecules.

Cat. No.

A10918

CAS No.

312753-06-3

Indacaterol

Synonyms: Arcapta; Onbrez

Indacaterol is an ultra-long-acting beta-adrenoceptor agonist.

Cat. No.

A11761

CAS No.

635701-59-6

Merck SIP Agonist

Cat. No.

A12288

CAS No.

105963-46-0

TOK-8801

TOK-8801 is a synthesized dihydroimidazothiazole carboxamide and is under development as an immunomodulator.

Cat. No.

A12594

CAS No.

1796641-10-5

Parimifasor

Synonyms: LYC30937

Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.

Cat. No.

A12908

CAS No.

1420071-30-2

Bioymifi

Bioymifi is a potent and selective small molecule agonist of DR5 that directly targets DR5, specifically binds the ECD of DR5 (Kd ~1.2 μM), and induces the formation of DR5 aggregates and DR5 activation.

Cat. No.

A13855

CAS No.

447407-36-5

AC-42 hydrochloride

Synonyms: AC 42

AC 42 is an allosteric agonist.

Cat. No.

A13960

CAS No.

259666-71-2

SM-130686

SM-130686 is a potent, orally active growth hormone secretagogue, with around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.

Cat. No.

A15334

CAS No.

481-42-5

Plumbagin

Plumbagin, exhibits cytotoxicity in rodent models of carcinogenesis and carcinoma; has antifungal, antiviral, and antibacterial action.

Cat. No.

A15852

CAS No.

220551-92-8

DAA-1106

Synonyms: DAA 110

DAA-1106 is a potent and selective ligand for peripheral benzodiazepine receptor (PBR), as a potent and selective agonist at the peripheral benzodiazepine receptor.

Cat. No.

A18880

CAS No.

2170608-82-7

PZ-2891

PZ-2891 is an orally bioavailable, brain penetrant pantothenate kinase (PANK) modulator. PZ-2891 act as an orthosteric inhibitor at high concentrations and an allosteric activator at lower sub-saturating concentrations. PZ-2891 inhibits human pantothenate kinases PANK1β, PANK2, and PANK3 with IC50s of 40.2 nM, 0.7 nM and 1.3 nM, respectively.