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Other Inhibitors

Other Inhibitors groups bioactive small molecules whose targets fall outside the pathway categories of this catalogue. The compounds have not yet been assigned to target categories, so the range is broad and uneven. Streptozotocin, a glucosamine-nitrosourea compound used to induce experimental diabetes in rodents, sits beside the O-GlcNAcase inhibitor Thiamet G. Exherin is an N-cadherin antagonist, and AdipoRon is an agonist of adiponectin receptors 1 and 2 (AdipoR1 and AdipoR2). Plant compounds such as the isoflavone daidzein are also included. Despite the category name, not every compound is an inhibitor, as the AdipoRon example shows. Compounds with a well-defined target are usually listed in the matching pathway or target category.

12 Items

  • UK-157147
    Cat. No.
    A12455
    CAS No.
    162704-20-3

    UK-157147

    UK-157147 is a substrate for UDP-glucuronosyltransferases (UGT1A1) with a Km value of 105 μM.

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    1 mg
    $200.00
    5 mg
    $500.00
    All 5 sizes
  • D-Luciferin
    Cat. No.
    A13789
    CAS No.
    2591-17-5

    D-Luciferin

    Synonyms: Firefly Luciferin

    D-Luciferin is a popular bioluminescent substrate of luciferase in the presence of ATP, used in luciferase-based bioluminescence imaging and cell-based high-throughput screening applications.

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    5 mg
    $30.00
    10 mg
    $40.00
    All 7 sizes
  • CPI-268456
    Cat. No.
    A15828
    CAS No.
    1380087-86-4

    CPI-268456

    CPI-268456 is a ligand of bromodomain-containing protein 4 (BRD4). It binds to BRD4 (IC50 =

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    1 mg
    $65.00
    5 mg
    $135.00
    All 4 sizes
  • CB1954
    Cat. No.
    A15862
    CAS No.
    21919-05-1

    CB1954

    Synonyms: Tretazicar

    CB1954 is a anticancer prodrug that is converted in the presence of the enzyme NQO2 and co-substrate caricotamide ( EP-0152R) (EP) into a potent cytotoxic bifunctional alkylating agent.It can be activated by NAD(P)H quinone oxidoreductase 2.

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    5 mg
    $40.00
    10 mg
    $65.00
    All 6 sizes
  • Coelenterazine
    Cat. No.
    A15897
    CAS No.
    55779-48-1

    Coelenterazine

    Synonyms: CLZN

    Coelenterazine is a luminescent enzyme substrate, used for monitoring reporter genes in BRET, ELISA and HTS techniques.

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    500 µg
    $60.00
    1 mg
    $90.00
    All 8 sizes
  • RETF-4NA
    Cat. No.
    A16019
    CAS No.
    1160928-63-1

    RETF-4NA

    RETF-4NA is a chymase substrate peptide that is cleaved more avidly by α2-macroglobulin-bound chymase than the free, unbound form.

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    1 mg
    $155.00
    5 mg
    $495.00
    All 2 sizes
  • DPA-714
    Cat. No.
    A18585
    CAS No.
    958233-07-3

    DPA-714

    Synonyms: J2.865.885K

    DPA-714 is a selective ligand for the translocator protein (TSPO) currently under evaluation for several clinical applications.It is also a PET tracer binding the TSPO receptor and highly expressed in myeloid cells.

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    1 mg
    $70.00
    5 mg
    $180.00
    All 8 sizes
  • 2'-Fluorothymidine
    Cat. No.
    A19148
    CAS No.
    122799-38-6

    2'-Fluorothymidine

    Synonyms: 2'-Deoxy-2'-fluoro-5-Methyluridine

    2'-Fluorothymidine (2'-Fluoro-2'-deoxythymidine), a bioisostere of both thymidine (TdR) and methyluridine, is a putative highly selective substrate for thymidine kinase type 2 (TK2).

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    1 mg
    $60.00
    5 mg
    $155.00
    All 7 sizes
  • BTTAA
    Cat. No.
    A20374
    CAS No.
    1334179-85-9

    BTTAA

    BTTAA is a Cu(I)-stabilizing ligand, whch performs potently with ubiquitin Glu18AzF.

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    1 mg
    $20.00
    5 mg
    $50.00
    All 6 sizes

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