PFI-2

Name: PFI-2
Brand: Adooq Bioscience
SKU: A14216
Rating: 5 (288 reviews)

Catalog No.: A14216

SETD7 inhibitor

PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibitor with Ki (app) and IC50 of 0.33 nM and 2 nM, 1000-fold selectivity over other methyltransferases and other non-epigenetic targets.

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Grouped product items
Size	Price	Stock
5mg	$75.00	In stock
10mg	$125.00	In stock
25mg	$230.00	In stock
50mg	$420.00	In stock
100mg	$800.00	In stock
*10mM 1mL in DMSO**	$105.00	In stock
Bulk Size	Bulk Discount

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Biological Activity

Description

Targets

Target	Value

Product Information

Catalog Num	A14216
Formula	C23H25F4N3O3S
Molecular Weight	499.52
CAS Number	1627676-59-8
SMILES	C1CCN(C1)C(=O)[C@@H](CC2=CC(=CC=C2)C(F)(F)F)NS(=O)(=O)C3=CC(=C4CNCCC4=C3)F
Synonyms	PFI2
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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