(S)-HH2853 is a potent dual inhibitor of EZH1 and EZH2, specifically targeting the EZH2_Y641F variant with an IC50 of less than 100 nM. This pyridine-based compound demonstrates significant biological activity, making it a valuable tool for research in anti-tumor and autoimmune disease pathways. Its ability to modulate histone methylation presents opportunities for exploring epigenetic regulation in various therapeutic contexts.
(S)-HH2853 is a potent dual inhibitor of EZH1 and EZH2, specifically targeting the EZH2_Y641F variant with an IC50 of less than 100 nM. This pyridine-based compound demonstrates significant biological activity, making it a valuable tool for research in anti-tumor and autoimmune disease pathways. Its ability to modulate histone methylation presents opportunities for exploring epigenetic regulation in various therapeutic contexts.
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