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Monoamine Transporter

Monoamine transporter inhibitors block reuptake of dopamine, noradrenaline and serotonin into neurons or vesicles. Plasma membrane transporters for dopamine (DAT), noradrenaline (NET) and serotonin (SERT) clear released transmitter from the synapse. Mice lacking DAT show hyperlocomotion and no response to cocaine or amphetamine, which identified this transporter as their main target. Vanoxerine 2HCl and GBR 12783 dihydrochloride are selective dopamine uptake inhibitors. Milnacipran hydrochloride inhibits both serotonin and noradrenaline reuptake at the plasma membrane. Vesicular monoamine transporters (VMAT) load monoamines into synaptic vesicles and are inhibited by reserpine. GZ-793A is a more selective inhibitor of the VMAT2 isoform.

2 Items

  • 2-(tert-Butylamino)-1-phenylpropan-1-one hydrochloride
    Cat. No.
    A67466
    CAS No.
    63199-74-6

    2-(tert-Butylamino)-1-phenylpropan-1-one hydrochloride

    2-(tert-Butylamino)-1-phenylpropan-1-one hydrochloride is a non-selective agonist of monoamine transporters, specifically targeting dopamine (DAT), norepinephrine (NET), and serotonin (SERT). This compound exhibits significant activity in modulating monoamine neurotransmission, making it a valuable tool for investigating the biochemistry underlying depressive disorders. It serves as a useful reagent in pharmacological studies aimed at understanding the mechanisms of mood regulation and potential therapeutic approaches.

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    Out of stock

    All 3 sizes
  • 4-MA-NBOMe hydrochloride
    Cat. No.
    A97273
    CAS No.
    2749298-47-1

    4-MA-NBOMe hydrochloride

    4-MA-NBOMe hydrochloride acts as a selective serotonin receptor agonist, specifically targeting the 5-HT2A receptor. This compound exhibits significant psychoactive properties and is utilized in neuroscience research to explore serotonergic signaling and its effects on behavior. Its activity in the amphetamine class makes it relevant for studies involving psychoactive substances and their neurological implications.

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    1 mg
    $105.00
    5 mg
    $330.00
    All 2 sizes

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