ZEN-2759 is a potent inhibitor of BET (bromodomain and extra-terminal domain) proteins, exhibiting IC₅₀ values of 0.23 μM for BRD4(BD1), 0.08 μM for BRD4(BD2), and 0.28 μM for BRD4(BD1BD2).
ZEN-2759 is a potent inhibitor of BET (bromodomain and extra-terminal domain) proteins, exhibiting IC₅₀ values of 0.23 μM for BRD4(BD1), 0.08 μM for BRD4(BD2), and 0.28 μM for BRD4(BD1BD2).
Product Information
Catalog Num
A24416
Formula
C17H16N2O2
Molecular Weight
280.32
CAS Number
1616400-50-0
SMILES
O=C1C=CC(C2=C(ON=C2C)C)=CN1CC3=CC=CC=C3
Storage
Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
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