dBRD4-BD1 is a selective BRD4 inhibitor that effectively induces degradation of the BRD4 protein, exhibiting a DC50 value of 280 nM (Dmax=77%). This compound not only selectively diminishes BRD4 levels but also promotes the upregulation of BRD2 and BRD3 protein levels, making it a valuable tool for studying the role of bromodomain proteins in cellular processes. Its low cytotoxicity profile compared to other BRD4 inhibitors highlights its potential for use in various research applications, including cancer biology and epigenetic regulation studies.
dBRD4-BD1 is a selective BRD4 inhibitor that effectively induces degradation of the BRD4 protein, exhibiting a DC50 value of 280 nM (Dmax=77%). This compound not only selectively diminishes BRD4 levels but also promotes the upregulation of BRD2 and BRD3 protein levels, making it a valuable tool for studying the role of bromodomain proteins in cellular processes. Its low cytotoxicity profile compared to other BRD4 inhibitors highlights its potential for use in various research applications, including cancer biology and epigenetic regulation studies.
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