EZH2-IN-22 is a potent inhibitor of EZH2, exhibiting IC50 values of less than 0.00051 µM for the EZH2 (Y641N) and EZH2 (Y641F) mutants, and 0.00052 µM for wild-type EZH2. This compound demonstrates significant antiproliferative activity, making it a valuable tool for research in epigenetic regulation and cancer biology. Its application extends to studies of EZH2-related pathways and therapeutic approaches for tumors exhibiting EZH2 mutations.
EZH2-IN-22 is a potent inhibitor of EZH2, exhibiting IC50 values of less than 0.00051 µM for the EZH2 (Y641N) and EZH2 (Y641F) mutants, and 0.00052 µM for wild-type EZH2. This compound demonstrates significant antiproliferative activity, making it a valuable tool for research in epigenetic regulation and cancer biology. Its application extends to studies of EZH2-related pathways and therapeutic approaches for tumors exhibiting EZH2 mutations.
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