I-BET282E is a selective pan-inhibitor of all eight BET bromodomains, effectively targeting BRD2, BRD3, and BRD4 with pIC50 values ranging from 6.4 to 7.7. This compound demonstrates potent inhibition and selectivity over other bromodomain-containing proteins, making it a valuable tool for investigating the role of BET proteins in cellular processes. I-BET282E is suited for research applications in cancer biology and epigenetic regulation.
I-BET282E is a selective pan-inhibitor of all eight BET bromodomains, effectively targeting BRD2, BRD3, and BRD4 with pIC50 values ranging from 6.4 to 7.7. This compound demonstrates potent inhibition and selectivity over other bromodomain-containing proteins, making it a valuable tool for investigating the role of BET proteins in cellular processes. I-BET282E is suited for research applications in cancer biology and epigenetic regulation.
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